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Competitive Information on GPCRs and GPCR Modulators
GPCR News	GPCR Google Search
	(Searches GPCR sites and companies)
GPCR modulator of the month: Adenosine A3 receptor agonists Gene Links: iHOP IUPHAR Biological significance: Receptor activation interrupts CD14 signaling and TNF induction Canfite CF101, RA, Dry Eye, Psoriasis (Phase II) Pipeline CF102, Liver Cancer, Hepatitis (Phase I) Pipeline CF502, Inflammation (Preclinical) Pipeline CV Therapeutics Research EP1537135A2; WO2003014137A1 Epigenesis Research EP1011608A2 King Research US6407236; US6448253; WO2005028489A2; WO2006055970A2 Muscagen Research WO2003061670A1 Pfizer Research US6921753 Trigen Research WO2005012323A2 US Gov Research WO2006031505A1
GPCR patents of the week (week ending May 30, 2008)
WO2008/063781 Abbott CB WO2008/064292 Abbott Nogo-66 US20080125425 Adenosine Therapeutics Adenosine A2 WO2008/064039 Allergan PG US20080125424 Amgen Ca sensing US20080125353 Amylin Exendin US20080125491 Arena GPCR US20080125435 Bayer-Schering EP2 US20080125463 Bayer-Schering EP2 US7378494 Bayer-Schering VPAC2 US7378418 BMS CB US7378409 BMS CCR2 WO2008/061966 Boehringer Ingelheim 5-HT2B WO2008/061968 Boehringer Ingelheim 5-HT2B WO2008/064054 Boehringer Ingelheim CB2 WO2008/062424 Cadila CB WO2008/062457 Cadila GLP-1 WO2008/062013 Cellzome Histamine H4 US7378098 Chemokine Thearapeutics CXCR4 WO2008/063600 Concert CCR5 WO2008/063712 CV Therapeutics Adenosine A2 WO2008/064202 Dr Reddys Ca Receptor US20080124742 Duke RTP US7378425 Eisai Sigma US20080125416 Esteve Sigma US20080125357 Euroscreen ChemerinR US20080125475 Grunenthal ORL1/Opioid mu US20080125422 GSK 5-HT4 WO2008/061955 GSK EP4 US20080124315 Individual CRF US20080124319 Individual MCH WO2008/063321 Jannssen GPR81 WO2008/064036 Jannssen Histamine H3 US20080125438 King Adenosine A1 WO2008/063984 King Adenosine A1 US7378447 Lilly Muscarinic M1 US7378448 Lilly Opioid US20080125468 Lilly Glucagon Receptor US20080125413 Merck CGRP US20080125443 Mount Cook Biosciences Delta Opioid US20080124384 Neurogen VR US20080125466 Neurogen VR US7378526 Neurosearch Nicotinic WO2008/061740 Novartis CXCR2 WO2008/061741 Novartis CXCR2 WO2008/062026 Novartis CXCR2 US7378500 Orthologic Thrombin Receptor WO2008/064351 Progenics Opioid WO2008/064353 Progenics    Opioid US20080125419 Roche Adenosine A2 WO2008/064338 Rubicon Angiotensin II US20080125461 Sepracor Leukotriene, Neurokinin, Adrenoceptor beta US7378524 Taigen CXCR3 WO2008/064310 Unic Med Dent NJ Opioid WO2008/064317 Unic Med Dent NJ Opioid WO2008/064318 Unic Med Dent NJ Opioid US7378385 Univ Cincinnati GLP-1 US7378400 Univ Virginia Adenosine 2A WO2008/064315 Univ Virginia Sphingosine 1 Phosphate WO2008/064320 Univ Virginia Sphingosine 1 Phosphate WO2008/064337 Univ Virginia Sphingosine 1 Phosphate WO2008/062296 Univ degli Stu de Ferrarra NOP US20080125455 Vernalis 5HT2C
Recent GPCR Reports   Market Opportunity in the G-Protein Coupled Receptors (GPCRs) Target Space: Qualitative and Quantitative Market Metrics Drug and Market Development 2007 $4,950.00 G-Protein Coupled Receptors 2007 Market Report Select Biosciences Limited Sep-2007 $3,535.00	GPCR links GPCR.org IUPHAR GPCR Database GPCR Natural Variants database   Upcoming GPCR Meetings
GPCR Books	GPCRs in Medicinal Chemistry 8-10 Sep 2008, Gothenburg, Sweden
All GPCR Books from Amazon
Companies working on GPCR modulators To be added

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